Identifying The Antagonists Receptor Hormone Inhibitor

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Endocrine therapy is the cornerstone of treatment for patients with hormone-receptor HR -positive advancedt cancer. In postmenopausal patients, aromatase inhibitors e.g., letrozole and anastrozole have become the treatment of choice in first-line therapy. 1-5 Unfortunately, not all patients have a response to first-line endocrine therapy .We report on the synthesis and biological evaluation of a series of 1,2-diarylimidazol-4-carboxamide derivatives developed as CB1 receptor antagonists. These were evaluated in a radioligand displacement bindin., a [35S]GTPS bindin., and in a compe.ionociationay that enables the relatively fast kinetic screening of .The insulin-like growth factor 1 IGF-1 receptor is a protein found on the surface of human cells.It is a transmem.ne receptor that is activated by a hormoneed insulin-like growth factor 1 and by a related hormoneed IGF-2.It belongs to the large clof tyrosine kinase receptors. This receptor mediates the effects of IGF-1, which is a polypeptide protein hormone .The cannabinoid type 1 receptor, often abbreviated as CB 1, is a G protein-coupled cannabinoid receptor located in the central and peripheral nervous system. It is activated by the endocannabinoid neurotransmitters anandamide and 2-arachidonoylglycerol ; by plant cannabinoids, such as the compound THC, an active ingre.nt of the .

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    A receptor antagonist is a type of receptor ligand or drug that blocks or dampens a biological response by binding to a receptor rather than prov.ng the response like an agonist.[1] They are sometimesed blockers; examples include alpha blockers, beta blockers, and calcium channel blockers..

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    Vasopressin antagonists are drugs that bind to vasopressin receptors V1A, V1B and V2 and block the action of vasopressin antidiuretic hormone, ADH , which is a hormone released by the pituitary gland..

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